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publicationNumber US-6967208-B2
titleOfInvention Lactam-containing compounds and derivatives thereof as factor Xa inhibitors
abstract The present application describes lactam-containing compounds and derivatives thereof of Formula I: or pharmaceutically acceptable salt forms thereof, wherein ring P, if present is a 5-7 membered carbocycle or heterocycle and ring M is a 5-7 membered carbocycle or heterocycle. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.
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Total number of triples: 5010.