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filingDate 2016-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-10-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6034883d759e866f48c5f4f810a39ceb
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publicationDate 2017-10-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9796766-B2
titleOfInvention Potent and selective inhibitors of NAV1.3 and NAV1.7
abstract Disclosed is a composition of matter comprising an isolated polypeptide, which is a peripherally-restricted Na V 1.7 inhibitor. In some disclosed embodiments, the isolated polypeptide is an inhibitor of Na V 1.7 and/or Na V 1.3. Other embodiments are conjugated embodiments of the inventive composition of matter and pharmaceutical compositions containing the inventive composition of matter. Isolated nucleic acids encoding some embodiments of inventive polypeptides and expression vectors, and recombinant host cells containing them are disclosed. A method of treating or preventing pain is also disclosed.
priorityDate 2011-03-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 2029.