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publicationNumber US-9744187-B2
titleOfInvention p-Ethoxy nucleic acids for liposomal formulation
abstract Provided herein are therapeutic oligonucleotides that comprise at least one p-ethoxy backbone linkage but no more than 80% p-ethoxy backbone linkages. Provided herein are improved delivery systems for therapeutic oligonucleotides comprising a liposome that comprises neutral phospholipids and a p-ethoxy oligonucleotide that is entrapped in the liposome.
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Total number of triples: 1144.