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publicationDate 2016-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9409892-B2
titleOfInvention 4-hydroxy-isoquinoline compounds as HIF hydroxylase inhibitors
abstract The present invention relates to novel compounds of formula (I), and compositions capable of inhibiting PHD1 enzyme activity selectively over other isoforms, for example, PHD2 and/or PHD3 enzymes. The invention also relates to compounds of formula (I) for use in disorders such as muscle degeneration, colitis, IBD, and certain ischemias.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID240222629
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226835401
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID224032776
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227168253
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431251082
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226571717
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89812933
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122443738
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID240222643
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431251051
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID240222649
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7971
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8785
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431251070
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226644078
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID240222688
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226457894
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89812929
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID240222692
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10868
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Total number of triples: 2409.