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filingDate 2011-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_704882a996f690dcac28c1c5696cf91d
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publicationDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9216995-B2
titleOfInvention Pyridone derivative having integrase inhibitory activity
abstract An object of the present invention is to provide a novel integrase inhibitor. The present invention relates to a novel compound having an antiviral effect, more specifically, a pyridone derivative having HIV integrase inhibitory activity, and a medicament containing the same, in particular, an anti-HIV agent. The compound of the present invention has integrase inhibitory activity and/or cell proliferation inhibitory activity against viruses, in particular, HIV and drug-resistant strains thereof. Thus, the compound is useful in preventing or treating various diseases, viral infections (for example, AIDS), and the like in which integrase participates.
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Total number of triples: 1317.