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publicationDate 2015-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9181245-B2
titleOfInvention Substituted pyrido[1,2-a]pyrazines and substituted pyrido[1,2-a][1,4]diazepines for the treatment of (inter alia) Alzheimer's disease
abstract The present invention is concerned with novel substituted 3,4-dihydro-2H-pyrido[1,2- a]pyrazine-1,6-dione derivatives of Formula (I) wherein R 1 , R 2 , R 3 , R 4 , R 5 , Z and X have the meaning defined in the claims. The compounds according to the present invention are useful as gamma secretase modulators. The invention further relates to processes for preparing such novel compounds, pharmaceutical compositions comprising said compounds as an active ingredient as well as the use of said compounds as a medicament.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503860
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413592916
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118073160
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18539871
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503859
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118073151
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118086203
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503858
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127812378
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118073149
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503849
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118073148
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503848
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426182067
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118073147
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454079093
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503847
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162181813
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118073155
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421757097
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118086324
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503846
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118073154
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118086256
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311503853
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID243859454
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22289852

Total number of triples: 3119.