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filingDate 2013-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-09-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_50e070c301ef7469dbb2b78b2681f878
publicationDate 2015-09-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9133126-B2
titleOfInvention Fluoroalkyl dibenzoazepinone compounds
abstract Disclosed are compounds of Formula (I): wherein R 1 is CH 2 CH2CF 3 or CH 2 CH2CH 3 ; R2 is CH 2 CH 2 CF 3 , CH 2 CH 2 CH 3 , CH 2 (cyclopropyl), phenyl, or; R 3 is H; R a , R b , y, and z are defined herein. Also disclosed are methods of using such compounds to inhibit the Notch receptor, and pharmaceutical compositions comprising such compounds. These compounds are useful in treating, preventing, or slowing the progression of diseases or disorders in a variety of therapeutic areas, such as cancer.
priorityDate 2012-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 872.