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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-14
filingDate 2012-10-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-05-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ff99fb13cf1815b358ea58f3a95c17d4
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_756a0948e66393cd7ab0b12d18e9cc48
publicationDate 2015-05-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9029364-B2
titleOfInvention 2,5-disubstituted thiomorpholine orexin receptor antagonists
abstract The present invention is directed to 2,5-disubstituted thiomorpholine amide compounds which are antagonists of orexin receptors. The present invention is also directed to uses of the 2,5-disubstituted thiomorpholine amide compounds described herein in the treatment or prevention of neurological and psychiatric disorders and diseases in which orexin receptors are involved. The present invention is also directed to pharmaceutical compositions comprising these compounds. The present invention is also directed to uses of these pharmaceutical compositions in the prevention or treatment of such diseases in which orexin receptors are involved.
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Total number of triples: 2325.