http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10017504-B2

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filingDate 2015-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-07-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_26bd93251cfc5ac5a578d5849529849d
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6720b1f0852b08ea8f3ca76148ec64b0
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publicationDate 2018-07-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10017504-B2
titleOfInvention Piperidine isoxazole and isothiazole orexin receptor antagonists
abstract The present invention is directed to piperidine isoxazole and isothiazole orexin compounds which are antagonists of orexin receptors. Such compounds are of the general structural formula I: n nwherein the variables are defined herein.n n The present invention is also directed to uses of the compounds described herein in the potential treatment or prevention of neurological and psychiatric disorders and diseases in which orexin receptors are involved. The present invention is also directed to compositions comprising these compounds. The present invention is also directed to uses of these compositions in the prevention or treatment of such diseases in which orexin receptors are involved.
priorityDate 2014-10-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 3005.