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grantDate 2013-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2013-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8524712-B2
titleOfInvention Triazinone and diazinone derivatives useful as HSP90 inhibitors
abstract The present invention relates to compounds according to formulae (IA) to (ID) and compositions that inhibit the activity of Hsp90. The invention further relates to methods of inhibiting the activity of Hsp90 in a subject in need thereof and methods for preventing or treating hyperproliferative disorders, such as cancer, in a subject in need thereof comprising administering to the subject a compound of the invention, or a composition comprising such a compound.
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Total number of triples: 4089.