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filingDate 2011-07-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b7d7c6cf28056fb07e46da0e1a00287e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_28cb4c1f4372228445c35497bfb90ee0
publicationDate 2013-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8513430-B2
titleOfInvention Substituted thiazol-2-ylamine derivatives, pharmaceutical compositions, and methods of use as 11-beta HSD1 modulators
abstract The present invention is directed to substituted thiazol-2-ylamine derivatives and pharmaceutically acceptable salts thereof that inhibit 11βHSD1 and that may be useful in the treatment of diseases in which modulation or inhibition of 11βHSD1 is beneficial or where a reduction in intracellular glucorticoid levels is desirable. The invention is also directed to pharmaceutical compositions comprising these compounds and the use of these compounds and compositions in the treatment of such diseases, disorders, or conditions in which modulation or inhibition of 11βHSD1 is beneficial or where a reduction in intracellular glucorticoid levels is desirable.
priorityDate 2010-07-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1787.