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filingDate 2006-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2012-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e40333bcc481e7d59b904ef68567234c
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publicationDate 2012-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8188288-B2
titleOfInvention 2-adamantylurea derivatives as selective 11beta-HSD1 inhibitors
abstract The present invention relates to 2-adamantylurea derivatives of formula I as selective inhibitors of the enzyme 11-beta-hydroxysteroid dehydrogenase type 1 (11β-HSD1) and the use of such compounds for the treatment and prevention of metabolic syndrome, diabetes, insulin resistance, obesity, lipid disorders, glaucoma, osteoporosis, cognitive disorders, anxiety, depression, immune disorders, hypertension and other diseases and conditions.
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Total number of triples: 858.