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filingDate 2006-11-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2011-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_80abbe5385fc9cc947406355cff111ea
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publicationDate 2011-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7947677-B2
titleOfInvention Spirolactam tricyclic CGRP receptor antagonists
abstract Compounds of formula I: n n(wherein variables A 1 , A 2 , A 3 , A 4 , A 5 , A 6 , A 7 , B 1 , B 2 , B 3 , B 4 , D 1 , D 2 , E 1 , E 2 , E 3 , E 4 , E 5 , G 1 , G 2 , J, K, T, U, V, W, X, Y and Z are as described herein) which are antagonists of CGRP receptors and which are useful in the treatment or prevention of diseases in which the CGRP is involved, such as migraine. The invention is also directed to pharmaceutical compositions comprising these compounds and the use of these compounds and compositions in the prevention or treatment of such diseases in which CGRP is involved.
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Total number of triples: 3433.