http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7659399-B2

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_b0128b1ea25bace77f9ff5dc6b2210d7
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-14
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D513-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4365
filingDate 2006-01-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2010-02-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f048c1f67bc0ba5fb1b1051f4ed49bc6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8e87fa2a0ee47378cfce27845aa56ca9
publicationDate 2010-02-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7659399-B2
titleOfInvention 1-thia-2,4a-diaza-cyclopenta[b]napththalene-3,4-diones and related compounds as anti-infective agents
abstract The invention provides compounds and salts of Formula I and Formula II: n nwhich possess antimicrobial activity. The invention also provides novel synthetic intermediates useful in making compounds of Formula I and Formula II. The variables A 1 , A 8 , R 2 , R 3 , R 5 , R 6 , R 7 , and R 9 are defined herein.n n Certain compounds of Formula I and Formula II disclosed herein are potent and selective inhibitors of bacterial DNA synthesis and bacterial replication. The invention also provides antimicrobial compositions, including pharmaceutical compositions, containing one or more compounds of Formula I or Formula II and one or more carriers, excipients, or diluents. Such compositions may contain a compound of Formula I or Formula II as the only active agent or may contain a combination of a compound of Formula I or Formula II and one or more other active agents. The invention also provides methods for treating microbial infections in animals.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2017197036-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2017197055-A1
priorityDate 2005-01-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 3101.