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filingDate 2002-09-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2009-05-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ba1106a0884b380a317fe99c844e72e4
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ec99a8a5386a798e6cdb1e57cb5c61a5
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publicationDate 2009-05-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7528162-B2
titleOfInvention 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity
abstract The present invention relates to a group of novel 4,5-dihydro-1H-pyrazole derivatives which are potent cannabinoid (CB 1 ) receptor antagonists with utility for the treatment of diseases connected with disorders of the cannabinoid system. The compounds have the general formula (I) wherein the symbols have the meanings given in the specification. The invention also relates to methods for the preparation of these compounds, and to pharmaceutical compositions containing one or more of these compounds as an active component.
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Total number of triples: 410.