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publicationDate 2007-06-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7230020-B2
titleOfInvention 11β-hydroxysteroid dehydrogenase inhibitors
abstract A compound having Formula In nR 1 —Z—R 2 Formula In nwherein R 1 is an optionally substituted phenyl ring; R 2 is or comprises an optionally substituted aromatic ring; and Z is —X—Y—L— or —Y—X—L— wherein either X is selected from —S(═O)(═O)— and —C(═O)—; and Y is —NR 3 —; or X is selected from —S(═O)(═O)— and —S—, and Y is —C(R 4 )(R 5 )—; L is an optional linker; and R 3 , R 4 and R 5 are each independently selected from H and hydrocarbyl; and wherein when R 2 comprises the following structural moietyn n nwherein Q is an atom selected from the group consisting of S, O, N and C; the compound is selected from compounds of the formulae R 1 —C(═O)—NR 3 —L—R 2 ; R 1 —S(═O)(═O)—C(R 4 )(R 5 )—L—R 2 ; R 1 —S—C(R 4 )(R 5 )—L—R 2 ; R 1 —NR 3 —S(═O)(═O)—L—R 2 ; R 1 —NR 3 —C(═O)—L—R 2 ; R 1 —C(R 4 )(R 5 )—S(═O)(═O)—L—R 2 ; and R 1 —C(R 4 )(R 5 )—S—L—R 2 .
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Total number of triples: 2413.