http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7026486-B2

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filingDate 2003-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2006-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6c53bd0b080764e5d1a3543ed33034ad
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publicationDate 2006-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7026486-B2
titleOfInvention Process for production cilostazol
abstract The present invention provides a process for producing cilostazol [I] in a high yield and a high purity, by reacting a carbostyril derivative [II] with a tetrazole derivative [III] in the presence of an inorganic basic compound in a solvent of water, wherein water is used in an amount of 3 to 7-fold weight to that of the carbostyril derivative [II] and the inorganic basic compound is used in an amount of 1 to 6 mol per mol of the carbostyril derivative [II]. The process of the present invention is the improved and environment-friendly process for producing cilostazol being useful for pharmaceuticals
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