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filingDate 2002-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2003-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a252db4133a550c6cba8a497e2e48228
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7d9787a53719cbb33e4be5a62f9e2449
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publicationDate 2003-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6642232-B2
titleOfInvention 3-[4-Substituted heterocyclyl)-pyrrol-2-ylmethylidene]-2- indolinone derivatives as kinase inhibitors
abstract The present invention relates to certain 3-[4-(substituted heterocyclyl)-pyrrol-2-ylmethylidene]-2-indolinone derivatives that inhibit kinases, in particular VEGFR and/or PDGFR kinases. Pharmaceutical compositions comprising these compounds, methods of treating diseases mediated by kinases utilizing pharmaceutical compositions comprising these compounds, and methods of preparing them are also disclosed.
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Total number of triples: 1871.