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filingDate 2000-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2002-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9cc3ef2c6b350dedee0feb21e95f49e7
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publicationDate 2002-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6423704-B2
titleOfInvention Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases
abstract The present invention relates to novel 4-(1H-benzimidazol-2-yl)[1,4]diazepane derivatives of formula (1):and stereoisomers thereof, and pharmaceutically acceptable salts thereof which are useful as histamine receptor antagonists and tachykinin receptor antagonist. Such antagonists are useful in the treatment of allergic rhinitis, including seasonal rhinitis and sinusitis; inflammatory bowel diseases, including Crohn's disease and ulcerative colitis; asthma; bronchitis; and emesis.
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Total number of triples: 4617.