http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-6403626-B1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_cc299202a8b5769ec9c8af124b3ac185 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-12 |
| filingDate | 2001-11-05-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2002-06-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5983774526a906ed159ec5167932e4ba http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c1ba4b2d5968c0c20623e266f4f9c371 |
| publicationDate | 2002-06-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | US-6403626-B1 |
| titleOfInvention | Benzimidazole derivatives |
| abstract | This invention provides compounds having the structure:wherein each of R1, R2, R3 and R9 is independently H; straight chain or branched, substituted or unsubstituted C1-C7 alkyl, C2-C7 alkenyl or alkynyl; C3-C7 cycloalkyl or cycloalkenyl; acyl, phenyl, substituted phenyl, or heteroaryl; wherein each dashed line represents a single bond or a double bond with the proviso that if R1 is present, R3 is absent and there is a double bond between N at position 3 and C at position 2 and a single bond between C at position 2 and N at position 1 and if R3 is present, R1 is absent and there is a double bond between N at position 1 and C at position 2 and a single bond between C at position 2 and N at position 3; wherein each of R4, R5 and R6 is independently H, F, Cl, Br, I; straight chain or branched, substituted or unsubstituted C1-C7 alkyl, C2-C7 alkenyl or alkynyl; C3-C7 cycloalkyl or cycloalkenyl; phenyl, substituted phenyl, heteroaryl, -OH, -OR7, -CN, -COR7, -CO2R7, -CON(R7)2, -OCOR7, -SR7, -N(R7)2, -NR7COR7, -(CH2)nOR7, -(CH2)nN(R7)2, -(CH2)nNR7COR7, wherein n is an integer from 1 to 4; and wherein each of R7 and R8 is independently H; straight chain or branched, substituted or unsubstituted C1-C7 alkyl, C2-C7 alkenyl or alkynyl; phenyl or substituted phenyl.These compounds are selective for cloned human alpha 2 receptors and are useful as analgesic, sedative or anaesthetic agents. |
| isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2218442-A1 |
| priorityDate | 1994-08-04-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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