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filingDate 1999-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2000-12-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2000-12-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6156339-A
titleOfInvention Process for preparing solid pharmaceutical dosage forms
abstract This invention relates to a process for the preparation of an oral solid rapidly disintegrating dosage form of a pharmaceutically active substance which has an unacceptable taste which process comprises: (i) forming a solution or a suspension in a solvent of a water soluble or water dispersible carrier, a filler and the pharmaceutically active substance with the unacceptable taste in association with a lipid, the weight ratio of the pharmaceutically active substance to the lipid being in the range of from 1:1 to 1:10 and the weight ratio of the carrier to the lipid being in the range of from 5:1 to 1:15; (ii) forming discrete units of the suspension or solution; and (iii) removing the solvent from the discrete units under conditions whereby unit dosages are formed comprising a network of carrier/filler carrying a dosage of the pharmaceutically active substance in association with the lipid; oral solid rapidly disintegrating dosage forms prepared by such a process are also provided.
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