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publicationDate 2000-07-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6083482-A
titleOfInvention Conformationally locked nucleosides and oligonucleotides
abstract Conformationally restricted 3',5'-bridged nucleoside analogues are described herein. The compounds can be prepared by cyclization at C3' and C5' of nucleosides through a linker or linking molecule. The nucleoside bases may be modified or unmodified. The nucleosides can be used as oligonucleotide building blocks or as small molecule pharmaceutical ingredients.
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