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filingDate 1999-05-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2000-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3a3be89787ed7a7bc557e52a4241d19f
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publicationDate 2000-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6054445-A
titleOfInvention Kappa agonist compounds pharmaceutical formulations and method of prevention and treatment of pruritis therewith
abstract Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics and anti-pruritic agents are provided. The compound of formulae IIA, having the structure: ##STR1## wherein R 1 , R 2 ; n X 4 , X 5 ; and n Ar and n are as described in the specification.
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Total number of triples: 4565.