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publicationDate 1999-04-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5891878-A
titleOfInvention Quinolones and their therapeutic use
abstract 1-Alkyl-substituted-quinolone-3-carboxamides have therapeutic utility via inhibition of Phosphodiesterase IV esterase and/or Tumour Necrosis Factor activity. The compounds of the invention have the general formula (I): ##STR1## The compounds of the invention encompassed by formula (I) include enantiomers, diastereoisomers and mixtures, including racemic mixtures.
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Total number of triples: 395.