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filingDate 1994-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1998-08-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5798332-A
titleOfInvention Glycosylation-mediated inhibition of factor X
abstract Reagents that specifically bind a carbohydrate target wherein sialic acid is linked at the nonreducing terminus of a glycoside to a galactose or galactosamine residue through an α2-6 linkage are able to inhibit the conversion of human Factor X to human Factor Xa. These reagents (SA/Gal/GalNAc binding reagents) as well as other strategies for inhibiting the conversion of Factor X to Factor Xa are useful in treating thrombosis, inflammation and other conditions associated with excess thrombin activity.
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