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publicationDate 1998-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5763445-A
titleOfInvention Kappa agonist compounds pharmaceutical formulations and method of prevention and treatment of pruritus therewith
abstract Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics and anti-pruritic agents are provided. The compounds of formular I, II, III and IV have the structure: <IMAGE> (I) <IMAGE> (II)X5, X7, X9; R1, R2, R3, R4; and Y, Z and n are as described in the specification.
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Total number of triples: 2499.