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filingDate 1993-03-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1997-10-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5679688-A
titleOfInvention Quinaldoyl-amine derivatives of oxo-and hydroxy-substituted hydrocarbons
abstract PCT No. PCT/AU93/00103 Sec. 371 Date Nov. 4, 1994 Sec. 102(e) Date Nov. 4, 1994 PCT Filed Mar. 11, 1993 PCT Pub. No. WO93/18006 PCT Pub. Date Sep. 16, 1993The present invention discloses the compounds of general formula (1) <IMAGE> wherein R1, R2, R3 are optionally substituted carbonyl and amide derivatives which are useful as inhibitors of retroviral proteases, and are effective in treating conditions characterized by unwanted activity of these enzymes, such as acquired immune deficiency syndrome.
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Total number of triples: 836.