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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3195517b064e87924b11bceaffb64c1e
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publicationDate 1994-03-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5296604-A
titleOfInvention Proline derivatives and compositions for their use as inhibitors of HIV protease
abstract The present disclosure describes novel peptidomimetic compounds which contain a novel class of isosteres and which inhibit the proteolytic activity of HIV protease and further describes therapeutic compositions comprising said compounds, a method of treatment for patients having the AIDS virus involving administering a therapeutically effective amount of the novel compounds of the present invention, and a method of preparation for said isosteres.
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