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publicationDate 1995-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5401747-A
titleOfInvention Alkyl camptothecin compounds as potent inhibitors of human colorectal cancer
abstract A method for synthesizing camptothecin and camptothecin analogs using a novel hydroxyl-containing tricyclic intermediate and the camptothecin analogs produced by the process. The camptothecin analogs are effective inhibitors of topoisomerase. I and show antileukemic and anti-tumor activity.
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