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publicationDate 1994-04-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5300674-A
titleOfInvention P2'-modified hydroxamic acid collagenase inhibitors
abstract Compounds of general formula I: ##STR1## Wherein: R 1 , R 2 , R 3 , R 4 , R 5 , and R 6 are variables. n These compounds have collagenase inhibition activity and are useful in the management of disease involving collagen degradation. Its uses include rheumatoide arthritis, corneal ulceration, osteoporosis, periodontitis, gingivitis and tumour invasion.
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Total number of triples: 429.