| abstract |
Aminophenylketone derivatives having excellent psychotropic activities and represented by the formula, WHEREIN R1 is hydrogen, C1-C4 alkyl or aryl; R is hydrogen or a group having the formula, -COR2 (wherein R2 is hydrogen, C1-C4 alkyl or aryl); R3 is hydrogen, halogen, C1-C4 alkyl, C1-C4 alkoxy or trifluoromethyl; R4 is hydrogen, C1-C4 alkyl or C1-C4 alkanoyl; R5 is C1-C4 alkyl or aryl; X is carbonyl or methylene; and Z is a group having the formula, (wherein R6 and R7 are each hydrogen, C1-C4 alkyl, aryl or aralkyl and R6 and R7 may form bivalent C2-C5 alkylene). |