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filingDate 2010-02-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_867efeae5216eb54ef2eab7a932ddab9
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publicationDate 2011-11-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2011288065-A1
titleOfInvention Aminopyrazine derivative and medicine
abstract The present invention relates to a compound represented by general formula [1] satisfying the following (I) or (II), or a pharmaceutical acceptable salt of the compound. n n n n n n n n n n (I) X is CH or N; R 1 is a halogen atom,; and R 2 is H, a halogen atom, CN, [2], [3], [8], [9], an —O-alkyl, an —O-(saturated ring), etc. n [2]: —C(R C )(R D )(R E ) (R C to R E each are H, an alkyl, etc.) n [3]: —N(R F )(R G ) (R F and R G each are H, OH, amino, a (hetero)aryl, etc.) n [8]: —C(═O)R L (R L is an alkyl, OH, an alkoxy, amino, etc.) n [9]: a (substituted)phenyl; n (II) X is >C—C(—O)R 3 (R 3 is a (substituted)amino, an alkoxy, OH, etc.); n R 1 is a halogen atom; R 2 is H; R 3 is H or OH; and R 3 and R 4 each are H or an alkyl.
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Total number of triples: 4575.