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filingDate 2008-11-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_33805e76fec188a4d5581d82ecf2846e
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publicationDate 2009-07-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2009175822-A1
titleOfInvention C5-substituted, proline-derived, macrocyclic hepatitis c serine protease inhibitors
abstract The present invention relates to compounds of Formula I or pharmaceutically acceptable salts, esters, or prodrugs thereof: n n n n n n n n n n which inhibit serine protease activity, particularly the activity of hepatitis C virus (HCV) NS3-NS4A protease. Consequently, the compounds of the present invention interfere with the life cycle of the hepatitis C virus and are also useful as antiviral agents. The present invention further relates to pharmaceutical compositions comprising the aforementioned compounds for administration to a subject suffering from HCV infection. The invention also relates to methods of treating an HCV infection in a subject by administering a pharmaceutical composition comprising a compound of the present invention.
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Total number of triples: 1491.