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filingDate 2008-01-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c9c3fedf7535e457a4f852d232570bed
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publicationDate 2008-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2008181868-A1
titleOfInvention Macrocylic oximyl hepatitis c protease inhibitors
abstract The present invention discloses compounds of formula I, or pharmaceutically acceptable salts, esters, or prodrugs thereof: n n n n n n n n n n which inhibit serine protease activity, particularly the activity of hepatitis C virus (HCV) NS3-NS4A protease. Consequently, the compounds of the present invention interfere with the life cycle of the hepatitis C virus and are also useful as antiviral agents. The present invention further relates to pharmaceutical compositions comprising the aforementioned compounds for administration to a subject suffering from HCV infection. The invention also relates to methods of treating an HCV infection in a subject by administering a pharmaceutical composition comprising the compounds of the present invention.
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Total number of triples: 1975.