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grantDate 2021-02-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_36afbee1c399e0e0b0fc67df76506804
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publicationDate 2021-02-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10919862-B2
titleOfInvention Fused imidazoles as mIDH1 inhibitors
abstract The present invention relates to compounds of general formula (I): in which R 1 , R 2 , R 3 , R 4 , R 6 , R 7 , R 8 , R 9 , R 10 , R 11 , R 12 , R 13 and X are as defined herein, to methods of preparing said compounds, to intermediate compounds useful for preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds and to the use of said compounds for manufacturing a pharmaceutical composition for the treatment or prophylaxis of a disease, in particular of neoplasms, as a sole agent or in combination with other active ingredients.
priorityDate 2015-07-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431962281
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419584834
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415810339
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396057

Total number of triples: 1891.