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publicationDate 2018-11-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10138226-B2
titleOfInvention Benzimidazol-2-amines as MIDH1 inhibitors
abstract The present invention relates to benzimidazol-2-amines of general formula (I) in which R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 , R 11 and R 12 are as defined herein, to methods of preparing said compounds, to intermediate compounds useful for preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds and to the use of said compounds for manufacturing a pharmaceutical composition for the treatment or prophylaxis of a disease, in particular of neoplasms, as a sole agent or in combination with other active ingredients.
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Total number of triples: 1785.