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titleOfInvention Derivatives of 5-(hetero)arylpyrazol-3-carboxylic amide or 1-(hetero)aryltriazol-4-carboxylic amide useful for the treatment of inter alia cystic fibrosis
abstract The present disclosure is based, in part, on the discovery that disclosed compounds such as those having Formula (IVa), (Va), (IV), or (V) can increase cystic fibrosis transmembrane conductance regulator (CFTR) activity as measured in human bronchial epithelial (hBE) cells.
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID379423
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID938861
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID829861
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419518689
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID179632
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24167359
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID422165
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397462
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A322
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID45124501
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18109
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08071
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56495
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6GKH9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8BFR4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453620572
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24338
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ29477
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP45376
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID554
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29219
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1023373
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID50018644
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393245
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07453
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ90744
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID230908
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100689318
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16220172
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4337720
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID62886811
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5143
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO59952
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100125267
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07489
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1023613
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397315
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID62886701
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID45051774
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID61129576
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD3ZQL7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP31779
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54670067
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8AAK6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07540
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8FAU3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD4A9L7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP45377
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6833
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP31955
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8615933
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJW7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ11129
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A287BM29
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID325052
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO64362
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJU0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID33037
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457493614
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID446948
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ48436
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30877
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJT9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID493887
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID449571
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1209619
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8018
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID31957
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6XQ98
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID947484
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID449649
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID40151856
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP50430
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID32051
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397150
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID62693680
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP50429
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280948
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ84177
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80276
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP76159
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID398723
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226415095
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ93MW7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280846
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23901
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9P4V4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24627
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14258306
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56419127
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396101
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID852721
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID294739
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP78285
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54676860
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID886174
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415272677
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A0E9

Total number of triples: 1052.