http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10660898-B2

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filingDate 2019-04-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-05-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8f4b29900e8b5f6880d7c06fa82505f9
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8414933a380ec264e559b64b05e7180d
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publicationDate 2020-05-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10660898-B2
titleOfInvention Benzimidazole derivatives as PI3 kinase inhibitors
abstract This invention relates to the use of benzimidazole derivatives for the modulation, notably the inhibition of the activity or function of the phosphoinositide 3′ OH kinase family (hereinafter PI3 kinases), suitably, PI3Kα, PI3Kδ, PI3Kβ, and/or PI3Kγ. Suitably, the present invention relates to the use of benzimidazoles in the treatment of one or more disease states selected from: autoimmune disorders, inflammatory diseases, cardiovascular diseases, neurodegenerative diseases, allergy, asthma, pancreatitis, multiorgan failure, kidney diseases, platelet aggregation, cancer, sperm motility, transplantation rejection, graft rejection and lung injuries. More suitably, the present invention relates to PI3Kβ selective benzimidazoles compounds for treating cancer.
priorityDate 2010-10-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415069749
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407121048
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452144692

Total number of triples: 1551.