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filingDate 2015-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6a58b9cbae45351f60743edb0e2dab79
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_14d445f4b12dda783b31958c78c5d6db
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publicationDate 2020-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10576064-B2
titleOfInvention Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitors
abstract The present invention relates to compounds of formula (I) n nwherein the groups R 1 to R 3 , R 7 , U, V, W, X, Y, n and q are as defined herein, their use as inhibitors of MDM2-p53 interaction, pharmaceutical compositions which contain compounds of this kind, their use as medicaments, especially as agents for treatment and/or prevention of oncological diseases and synthetic intermediates.
priorityDate 2014-07-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 2401.