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publicationDate 2019-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10508101-B2
titleOfInvention Protein kinase C inhibitors and methods of their use
abstract PKC inhibitors are disclosed. The PKC inhibitors are useful for treating PKC associated diseases, including certain cancers. The PKC inhibitors have improved efficacy at lower dosage amounts to achieve tumor regression, improved potency, PK profile, absorption, gastrointestinal tolerance and kinase selectivity.
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Total number of triples: 525.