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filingDate 2016-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-01-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2019-01-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10167266-B2
titleOfInvention Sodium channel blockers
abstract The present invention relates to compounds of Formula (I) and pharmaceutical compositions thereof. Compounds of Formula (I) are epithelial sodium channel (ENaC) blockers useful in the hydration of mucosal surfaces, enhancement of mucociliary clearance, or restoration of mucosal defense in a subject. The compounds and compositions can therefore be used to treat diseases which rely on the hydration of mucosal surfaces.
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Total number of triples: 1163.