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filingDate 2017-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-07-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_53aca7a9db12e15b5515abf55fdde507
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publicationDate 2018-07-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10018619-B2
titleOfInvention Compounds and method of identifying, synthesizing, optimizing and profiling protein modulators
abstract This invention relates to methods of identifying, synthesizing, optimizing and profiling compounds that are inhibitors or activators of proteins, both naturally occurring endogenous proteins as well as certain variant forms of endogenous proteins, and novel methods of identifying such variants. The method accelerates the identification and development of compounds as potential therapeutically effective drugs by simplifying the pharmaceutical discovery and creation process through improvements in hit identification, lead optimization, biological profiling, and rapid elimination of toxic compounds. Implementation results in overall cost reductions in the drug discovery process resulting from the corresponding increases in efficiency.
priorityDate 2005-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID230335359
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161450706
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID416939
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51445
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162094231
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID425792
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450108871
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C781
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID558154
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58876829
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51567
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158829633
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51568
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID340418773
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58876840
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51566
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Total number of triples: 3597.