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filingDate 2014-03-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-06-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_099b291f596bf82a8ccbe052f2e88aa3
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publicationDate 2018-06-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2656597-C2
titleOfInvention Quinazoline inhibitors of activating mutant forms of epidermal growth factor receptor
abstract FIELD: chemistry. n SUBSTANCE: invention relates to organic chemistry, specifically a heterocyclic compound of formula (I) or a pharmaceutically acceptable salt thereof. Invention also relates to a pharmaceutical composition based on a compound of formula (I) or a pharmaceutically acceptable salt thereof, use thereof and a method of treating cancer. . n EFFECT: technical result: obtaining a novel compound of formula (I) and pharmaceutically acceptable salts thereof, having inhibitory activity with respect to activating mutated forms of EGFR and useful in the treatment of cancer. n 16 cl, 10 tbl, 12 dwg, 7 ex
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