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filingDate 2003-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_14938dd519b9a442c5ee65921f0bf3a1
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6d607b8cfa82e79000193712e741b9e4
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_994087fbb6b982973bc2988f93510c3f
publicationDate 2007-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EA-009300-B1
titleOfInvention 4- (N-PHYLENAMINO) QUINAZOLIN / -CHINOLINE AS THYROSINKINASE INHIBITORS
abstract The invention describes bicyclic heterocycles of general formula (I) in which R, R, R, R and X have the meanings indicated in claim 1, their tautomers, their stereoisomers, their mixtures and their salts, especially their physiologically compatible salts with inorganic or organic acids, while such compounds have valuable pharmacological properties, primarily the inhibitory effect on signal transduction mediated by tyrosine kinases, and the use of these compounds for the treatment of various diseases, primarily of neoplastic diseases, as well as benign prostatic hyperplasia, diseases of the lungs and airways, and the preparation thereof.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2656597-C2
priorityDate 2002-03-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 579.