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filingDate 2010-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2017-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-101766931-B1
titleOfInvention Method for producing methyl-(4,6-diamino-2-(1-(2-fluorobenzyl)-1h-pyrazolo(3,4-b)pyridino-3-yl)pyrimidino-5-yl)methylcarbamate and its purification for use thereof as pharmaceutical substance
abstract The present invention relates to a process for the preparation of methyl- {4,6-diamino-2- [1- (2-fluorobenzyl) -1H-pyrazolo [3,4- b] pyridino- Pyrimidino-5-yl} methylcarbamates and for the purification of crude products of compounds of formula (I) for use as pharmaceutical active substances. For purification, methyl- {4,6-diamino-2- [1- (2-fluorobenzyl) -1H-pyrazolo [3,4- b] pyridino- -Yl} methylcarbamate-sulphonyldimethan (1: 1), i.e. a compound of formula (II) below, is isolated as an intermediate present in the mixture optionally in the purification process or is produced as an intermediate. &Lt; Formula (I) > &Lt; Formula (II) >
priorityDate 2009-11-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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