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filingDate 2018-01-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-06-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2020518240-A
titleOfInvention An endolysosomal targeting conjugate for enhanced delivery of cargo molecules to the endolysosomal compartment of target cells
abstract Explaining endolysosomal targeting conjugates modified to deliver cargo molecules such as cytotoxic drugs or imaging labels to late endosomes and/or lysosomes in target cells such as tumor cells with improved efficiency .. The endolysosomal targeting conjugate comprises a targeting component and a cargo component. The targeting component is configured to bind to a cell surface molecule of a target cell and the cargo component comprises a cargo molecule. The targeting moiety and cargo moiety may be covalently fused or non-covalently associated. The targeting moiety may bind to a cell surface molecule or cargo moiety in the extracellular space with a higher affinity in the endolysosomal compartment of the target cell. [Selection diagram] Figure 1
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100005148
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9848990
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21251
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID213
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14187
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46096
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID337132
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18061
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3T0L5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ15075
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ60HC0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48018
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6857
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419487901
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24044
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24551
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID386966
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID247744
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100009195
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07463
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11657
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20692
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48036
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID39130
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCG3V226
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29183
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47191
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04083
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5U4Z2
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID9838
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419484124
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24329
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100009122
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6XQ98
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4332664
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06731
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51728
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13075
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24186
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04464
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92108
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24208
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID451185
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID69538
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID282077
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24192
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2346
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO55159
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11677
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448484808
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04352
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12478
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID101152771
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID35411
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A2R8QP29
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17967
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID84168
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412568307
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419521378
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13559
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09963
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID216238
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6453725
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04353
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5R4J5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A1D5PWY3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15094
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID85302
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8728
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID85309
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO82018
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9793
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24586
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12494
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16952
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2064
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24926
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO64362
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396816
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17075
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396494
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP14668
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62693
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ99JW5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ71UH5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9832481
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9U6D3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41823
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5175
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8N158
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61859
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419529789
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ71UH6

Total number of triples: 414.