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filingDate 2015-12-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2017-12-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2017536401-A
titleOfInvention Anticancer composition
abstract The present invention relates to pharmaceutical formulations of ARN-509, which formulations are androgen receptor (AR) related diseases or conditions, specifically cancer, more specifically prostate cancer, such as, but not limited to, Castration-resistant prostate cancer, metastatic castration-resistant prostate cancer, chemotherapy-naïve metastatic castration-resistant prostate cancer, biochemically recurrent hormone-sensitive positive prostate cancer, or high-risk non-metastatic castration-resistant prostate cancer Can be administered to mammals, particularly humans. In one aspect, these formulations comprise a solid dispersion of ARN-509 and a poly (meth) acrylate copolymer. In one aspect, a solid dispersion of ARN-509 and poly (meth) acrylate copolymer is melt extruded from a mixture comprising ARN-509 and poly (meth) acrylate copolymer, optionally followed by It is obtainable, in particular obtained, by grinding the melt-extruded mixture. In one aspect, the solid dispersion of ARN-509 and poly (meth) acrylate copolymer is spray dried from a mixture comprising the mixture comprising ARN-509 and poly (meth) acrylate copolymer in a suitable solvent. And is particularly obtainable.
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