http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2016519059-A

Outgoing Links

Predicate Object
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-12
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-16
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D205-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-16
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K7-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K7-08
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K1-113
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K1-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K7-50
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P15-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P1-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K1-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P1-16
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K1-10
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P11-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P7-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P5-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P37-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P29-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K38-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-16
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D205-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K7-54
filingDate 2014-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-06-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016519059-A
titleOfInvention Stapled and stitched polypeptides and uses thereof
abstract The present invention provides stapled polypeptides of formulas (I) and (VI), (I) (VI) and salts thereof, wherein the group , R 1a , R 1b , R 1c , R 2a , R 3a , R 2b , R 3b , R 4a , R 4b , R A , R Z , L 1a , L 1b , L 2 , L 3 , X AA , v , W, p, m, s, n, t, and q are as defined in this application. The present invention further provides methods for preparing the stapled polypeptides of the present invention from non-staple polypeptide precursors. The present invention further provides pharmaceutical compositions comprising a stapled polypeptide of formula (I) or (VI), and methods of using the stapled peptide. The present invention also provides for the modification of staples after ring closure metathesis.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-7361689-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2020528458-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2020533413-A
priorityDate 2013-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2008501623-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2011156686-A2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2012065181-A2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2008242598-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2010510236-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2010522769-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2012532929-A
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID78632
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID183277
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID4232
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466892936
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID39329
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID51089
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID13363
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID48032
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID69008
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID35974
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70059
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID4146
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97399
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID51240
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7TQD2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396200
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID8010
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID51089
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID452646
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID1878969
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID69008
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID4443
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID8010
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467123989
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID39343
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466717038
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17246
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466718854
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35049
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID1878969
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35050
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID3999
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID492274
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35051
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9VV43
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD3ZQL7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4193
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID295139
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395609
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID8790
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID99037
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID8790
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO94811
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID30637
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID175205
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00761
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID9541
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID30590
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID314856
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID3755
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID349346
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397926
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID51240
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID492274
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID452646
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID193516
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID512563
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID3663
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID180016
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ27957
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID4222
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83348
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281542
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID270329
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID180016
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403693
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID9544
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID742141
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID292385
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19799
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID183277
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID262690
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID13363
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID167337
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467104012
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID48032
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9544
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24664
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID34318
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID852825
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID3435
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID22059
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00764
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID262690
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397276
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403869
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00775
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID12721
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466090063
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID4146
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID35974
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID49987
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID3999
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID36596
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID193516
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID540378
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID27787
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID1053382
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID4443
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID39343
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID295139
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID49987
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81071
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID27787
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID39367
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID3435
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466148573
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID34318
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59149
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID36596
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID39367
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID4232
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID8049
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID455214
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23916
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100379269
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467772729
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID349346
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID3755
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467773126
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7157
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24842
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID128608
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID99037
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID4222
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID78632
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID270329
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID175205
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID128608
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID3663
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35034
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35048
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID292385
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID12721
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID167337
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466869265
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID39329
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51588
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID512563
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID1053382
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID8049

Total number of triples: 202.