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filingDate 2012-07-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2014-08-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2014520848-A
titleOfInvention Process for the preparation of type 1 fluticasone propionate
abstract The present invention relates to a novel crystallization method for preparing fluticasone propionate as a type 1 polymorph crystal having a controlled particle size and suitable for micronization. The method involves dissolving fluticasone propionate in acetone or a mixture of acetone and water, and then adding the solution to water or a mixture of water 10 and acetone, whereby fluticasone propionate is crystallized from the solution. A step of causing crystallization in the form. [Selection] Figure 4
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