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filingDate 2010-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2012-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2012522732-A
titleOfInvention Piperidine and piperazine derivatives as autotaxin inhibitors
abstract The present invention is caused and mediated by piperidine and pyrazine derivatives according to formulas (Ia), (Ib) and (II) as autotaxin inhibitors, and increased lysophosphatidic acid levels and / or activation of autotaxin, It relates to the use of such compounds for the treatment and / or prevention of and / or amplified physiological and / or pathophysiological conditions, in particular various cancers.
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priorityDate 2009-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB3W9W2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5CCC1
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5SJ26
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5Z8N5
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8RDT4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0JH94
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5IM27
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3AQS4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5X3L5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1QRF9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ57FA3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6L8E5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1QRY3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24835
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID317748
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9MRU6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5N2H7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4FUF9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ60BT7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5IDM1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ89WP0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0ABM5
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2RN87
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12IW9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8KDS1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ253S7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2I858
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6L391
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO67613
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2RL24
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ38YR2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ89V00
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ817R9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2JNH4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1AVT5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3KM09
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID3704
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8RFE6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Z9F9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2C7X9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ21CL6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ72ZX1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7TWT7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18605
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8RBC6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ49670
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ82I23
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18606
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4UJ23
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8FA20
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ87EA3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396816
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05205
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5QWE2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11839
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A749
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0AKD7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ88PB4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1CS23
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ73K74
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ73KL7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12367
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID562399
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12C38
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100126739
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC6E559
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395476
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11835
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ73I47
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2G9H1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7GHM0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5G7S1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9AC58
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8F031
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2C3V6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID747460
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2GC58
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4XKL5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID36054
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3L6Y6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9K8H3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VB43
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1IV55
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ989F1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0TCL8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP25536
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ15ZH0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16101
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0AWG2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7NH22
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ63VT5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8FFU1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4SA80
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3IYH0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3P9E0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ57J97
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9PI04
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID494527
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1DAV2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13075
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8XIH4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GXY9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ04XA6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3J086
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ02169
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ39X87
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423796612
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9ZCE2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4ZDP0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3L3L1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6JN80
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2RQN0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1D912
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8P7K1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8L0X4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3YRV1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0HEI2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05700
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GTV6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13487
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5FGZ7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13254
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6QP91
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2JXB4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0S919
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1I4S1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5NNS3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO59604
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ73UG7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VKR7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7GTD6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416164029
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ67SI8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID422165
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID3704
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID374
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8U476
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7U5K1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5FA52
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1NNP2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO84353
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6LJI7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2S4I1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3J7T5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9KHL6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4JTL6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2GKV0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100689061
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0AQL3
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID11103
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1UCG3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GQ13
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ81LD6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ66I23
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0YX95
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3AWW1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2GGV6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ665F6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2W1Y3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9NE14
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6N181
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1BCI0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5L6G5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8HN65
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58056893
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ169N3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5167
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5D426
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8E0U2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID36203
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5168
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2UPE6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0SK44
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ315F5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0ZWV2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1R741
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3PW53
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5N6I4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2GCP9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1IYX1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3PLU6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8DCG8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ82ZA4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2KCN4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6LQP7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ12TU6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7IIW6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11997
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ68VT4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3YX01
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ47JQ0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2VYH3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3JUG5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5Z154
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9ZJY6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1LQB1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3PEA3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6A725
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81800
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7IFS5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5D5H8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7MHE0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0B7R8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2YC50
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1R692

Total number of triples: 608.